CYN 154806 (TFA), a cyclic octapeptide, is a potent and selective somatostatin sst2 receptor antagonist, with pIC50 values of 8.58, 5.41, 6.07, 5.76 and 6.48 for human recombinant sst2, sst1, sst3, sst4 and sst5 receptors respectively.
CAT# | R1320 |
M.F/Formula | C₅₈H₆₉F₃N₁₂O₁₆S₂ |
M.W/Mr. | 1311.36 |
Sequence | One Letter Code: Ac-Phe-Cys-Tyr-Trp-Lys-Thr-Cys-Tyr-NH2 (Disulfide bridge: Cys2-Cys7) three Letter Code: Ac-FCYWKTCY-NH2 (Disulfide bridge: Cys2-Cys7) |
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