Difelikefalin ,also known as D-Phe-D-Phe-D-Leu-D-Lys-[γ-(4-N-piperidinyl)amino carboxylic acid] (as the acetate salt), is an analgesic opioid peptide acting as a peripherally specific, highly selective agonist of the κ-opioid receptor (KOR).
CAT# | 10-101-174 |
CAS | 1024828-77-0(net);1024829-44-4 |
Synonyms/Alias | CR845 acetate;CR-845 acetate;UNII-0P70AR5BYB; 0P70AR5BYB; |
M.F/Formula | C38H57N7O8 |
M.W/Mr. | 739.90128 |
Labeling Target | K-opioid receptor |
Application | Difelikefalin is an intravenous agent for the treatment of postoperative pain. |
Activity | Agonist |
Biological Activity | Difelikefalin acetate is a kappa opiate receptor agonist that is used for its antipruritic effects. |
Areas of Interest | Postoperative pain |
Disease | Acute Pain and Postoperative Pain |
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