GPS1573 Peptide

GPS1573 is a newly described potent and dose-dependent peptide antagonist of ACTH-stimulated melanocortin type 2 receptor (MC2R) activity in vitro (IC50 = 66 nM). GPS1573 antagonizes MC4R with IC50 of 950 nM, therefore showing selectivity for MC2R. The binding of ACTH to MC2R regulates steroidogenesis leading to metabolic diseases such as Cushing's disease in patients with pituitary dysfunctions.

Online Inquiry

Specification Technical Data Related Products Featured Products Customer reviews and Q&A Useful Tools Publications

CAT#	A03042
Synonyms/Alias	GPS1573; MC2R antagonist; Adrenocorticotropic hormone receptor antagonist
M.F/Formula	C86H139N27O16
M.W/Mr.	1807
Sequence	Three-Letter Code: H-Nle-Pro-(D-Phe)-Arg-(D-Trp)-Phe-Lys-Ala-Val-Gly-Lys-Lys-Arg-Arg-NH2 One-Letter Code: H-Nle-PfRwFKAVGKKRR-NH2
Purity	Purity > 95% by HPLC

CAT#	Product Name	Inquiry
A03040	Sauvagine	Inquiry
A03012	Acetyl-ACTH (3-24) (human, bovine, rat)	Inquiry
A03006	(Tyr15)-ACTH (7-15)	Inquiry
A03021	ACTH (12-39), rat	Inquiry
A03045	(D-Ser¹)-ACTH (1-24) (human, bovine, rat) trifluoroacetate salt	Inquiry

CAT#	Product Name	M.W	Molecular Formula	Inquiry
10-101-20	Goserelin Acetate	1269.43	C59H84N18O14	Inquiry
10-101-59	Liraglutide	3751.2	C172H265N43O51	Inquiry
R1574	Octreotide	1019.24	C₄₉H₆₆N₁₀O₁₀S₂	Inquiry
10-101-139	Myrcludex B			Inquiry
10-101-285	Teduglutide	3752.08	C164H252N44O55S	Inquiry
R1847	Sermaglutide	4114	C187H291N45O59	Inquiry
R1961	Carbetocin	988.2	C45H69N11O12S	Inquiry

If you have any peptide synthesis requirement in mind, please do not hesitate to contact us at . We will endeavor to provide highly satisfying products and services.

Length	7
Storage	Store at -20°C. The product is hygroscopic and must be protected from light. Product is guaranteed one year from the date of shipment. Following reconstitution, aliquot and store at -20°C.