Potent human MC1 receptor antagonist (IC50 = 17 nM), and alsoMC3 and MC5 partial agonist (EC50 values are 59 and 1300 nM, respectively). Exhibits binding affinity for A375 melanoma.
CAT# | R1043 |
CAS | 1416983-77-1 |
M.F/Formula | C62H82N20O13S |
M.W/Mr. | 1347.51 |
Sequence | XGHFRWCDRFG(Modifications: X = Butanoic acid, Gly-11 = C-terminal amide, Phe-4 = D-Phe, Trp-6 = D-Trp, carba sulfide bridge between X-1 - Cys-7) |
Labeling Target | MC1 receptor |
Activity | Antagonist |
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