Bremelanotide, formerly known as PT-141, is a peptide drug. Bremelanotide acts as a non-selective agonist of all of the melanocortin receptors except MC2.
CAT# | 10-101-112 |
Chemical Structure | |
CAS | 189691-06-3 |
Synonyms/Alias | (Ac-Nle4, Asp5, D-Phe7, Lys10)-cyclo-α-MSH (4-10); PT-141; PT 141; PT141 |
Chemical Name | (3S,6S,9R,12S,15S,23S)-15-[[(2S)-2-acetamidohexanoyl]amino]-9-benzyl-6-[3-(diaminomethylideneamino)propyl]-12-(1H-imidazol-5-ylmethyl)-3-(1H-indol-3-ylmethyl)-2,5,8,11,14,17-hexaoxo-1,4,7,10,13,18-hexazacyclotricosane-23-carboxylic acid |
M.F/Formula | C50H68N14O10 |
M.W/Mr. | 1025.18 |
Sequence | Three Letter Code: Ac-Nle-cyclo(-Asp-His-D-Phe-Arg-Trp-Lys);Ac-Nle-cyclo(-Asp-His-D-Phe-Arg-Trp-Lys)-OH |
Application | Erectile dysfunction & Female sexual dysfunction & Hemorrhagic shock & Reperfusion injury |
Appearance | White Powder |
Activity | Agonist |
Target | Melanocortin Receptor |
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