Selective and competitive silent antagonist for the NOP opioid receptor that binds to NOP with high affinity (pKi = 10.24) and displays > 3000-fold selectivity over δ, μ and κ opioid receptors.
CAT# | R1067 |
CAS | 849024-68-6 |
Synonyms/Alias | [Nphe1,Arg14,Lys15]Nociceptin-NH2 |
M.F/Formula | C82H138N32O21 |
M.W/Mr. | 1908.19 |
Sequence | GGGFTGARKSARKRKNQ(Modifications: Gly-1 = N-(Bn)Gly, Gln-17 = C-terminal amide) |
Labeling Target | NOP opioid receptor |
Appearance | White lyophilised solid |
Purity | >98% |
Activity | Antagonist |
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