Targeting Peptides

Designed for biological research and industrial applications, not intended for individual clinical or medical purposes.
Name CAS MF MW Single-letter sequence Three-letter sequence Number of AA Type Inquiry
TPP-1 C107H150N34O32S2 2488.67 H2N-SGQYASYHCWCWRDPGRSGGSK-OH H2N-Ser-Gly-Gln-Tyr-Ala-Ser-Tyr-His-Cys-Trp-Cys-Trp-Arg-Asp-Pro-Gly-Arg-Ser-Gly-Gly-Ser-Lys-OH 22 PD-L1–targeting peptide
HAC-V C49H80N14O14 1089.24 H2N-HVVHEGTVVI-OH H2N-His-Val-Val-His-Glu-Gly-Thr-Val-Val-Ile-OH 10 PD-L1–targeting peptide
DPPA-1 C70H98N20O21 1555.65 H2N-nyskptdrqyhf-OH H2N-DAsn-DTyr-DSer-DLys-DPro-DThr-DAsp-DArg-DGln-DTyr-DHis-DPhe-OH 12 PD-L1–targeting peptide
AP-1 C107H150N34O32S2 2488.67 H2N-SGQYASYHCWCWRDPGRSGGSK-OH H2N-Ser-Gly-Gln-Tyr-Ala-Ser-Tyr-His-Cys-Trp-Cys-Trp-Arg-Asp-Pro-Gly-Arg-Ser-Gly-Gly-Ser-Lys-OH 22 APN-targeting peptide
EP-1 C49H80N14O14 1089.24 H2N-HVVHEGTVVI-OH H2N-His-Val-Val-His-Glu-Gly-Thr-Val-Val-Ile-OH 10 EpCAM-targeting peptide
GSC-IC2 C51H58N8O11 959.05 H2N–AWEFYFP–OH H2N–Ala–Trp–Glu–Phe–Tyr–Phe–Pro–OH 7 GBC tumor–targeting peptide
STP C70H98N20O21 1555.65 H2N-nyskptdrqyhf-OH H2N-DAsn-DTyr-DSer-DLys-DPro-DThr-DAsp-DArg-DGln-DTyr-DHis-DPhe-OH 12
RES-701-1 151308-34-8 C103H115N23O23 2043.19 Cyclo(-GNWHGTAPD)WFFNYYW Cyclo(-Gly-Asn-Trp-His-Gly-Thr-Ala-Pro-Asp)-Trp-Phe-Phe-Asn-Tyr-Tyr-Trp-OH 16
SYLQDSVPDSFQD 320341-56-8 C65H93N15O26 1500.52 H2N-SYLQDSVPDSFQD-OH H2N-Ser-Tyr-Leu-Gln-Asp-Ser-Val-Pro-Asp-Ser-Phe-Gln-Asp-OH 13
Thrombospondin-1 (TSP-1)–derived CD36 Binding Motif 138849-26-0 C20H34N6O9S2 566.65 H2N-CSVTCG-OH H2N-Cys-Ser-Val-Thr-Cys-Gly-OH 6
ELT C60H90N12O19S2 1347.56 H2N-ELTVMGYYPGMS-OH H2N-Glu-Leu-Thr-Val-Met-Gly-Tyr-Tyr-Pro-Gly-Met-Ser-OH 12 Gastric cancer–targeting peptide
GLP-1(28-36)amide 1225021-13-5 C54H85N15O9 1088.35 H2N-FIAWLVKGR-CONH2 H2N-Phe-Ile-Ala-Trp-Leu-Val-Lys-Gly-Arg-CONH2 9 Mitochondria-targeting peptide
CBO-P11 612096-46-5 C94H145N29O25S 2113.4 Cyclo(RIKPHQGQHIGEDFPQIM) Cyclo(Asp-Phe-Pro-Gln-Ile-Met-Arg-Ile-Lys-Pro-His-Gln-Gly-Gln-His-Ile-Gly-Glu) 18 Tumor Angiogenesis-targeting ligands
TAT-GluN2BCTM 1587742-50-4 C224H374N86O54 5135.91 H2N-YGRKKRRQRRRKKNRNKLRRQHSYKFERQKILDQRFFE-OH H2N-Tyr-Gly-Arg-Lys-Lys-Arg-Arg-Gln-Arg-Arg-Arg-Lys-Lys-Asn-Arg-Asn-Lys-Leu-Arg-Arg-Gln-His-Ser-Tyr-Lys-Phe-Glu-Arg-Gln-Lys-Ile-Leu-Asp-Gln-Arg-Phe-Phe-Glu-OH 38 DAPK1–targeting peptide
KGYY15 1690215-31-6 C84H129N21O22S1 1815.93 H2N-VLQWAKKGYYTMKSN-OH H2N-Val-Leu-Gln-Trp-Ala-Lys-Lys-Gly-Tyr-Tyr-Thr-Met-Lys-Ser-Asn-OH 15 CD40–targeting peptide
TPP-1 C107H150N34O32S2 2488.67 H2N-SGQYASYHCWCWRDPGRSGGSK-OH H2N-Ser-Gly-Gln-Tyr-Ala-Ser-Tyr-His-Cys-Trp-Cys-Trp-Arg-Asp-Pro-Gly-Arg-Ser-Gly-Gly-Ser-Lys-OH 22 PD-L1–targeting peptide
HKP2201 C77H101N21O20 1640.75 H2N–WHRSYYTWNLNT–OH H2N–Trp–His–Arg–Ser–Tyr–Tyr–Thr–Trp–Asn–Leu–Asn–Thr–OH 12 PD-L1–targeting peptide
EDIKPKTSLAFR C63H105N17O19 1404.61 H2N-EDIKPKTSLAFR-OH H2N-Glu-Asp-Ile-Lys-Pro-Lys-Thr-Ser-Leu-Ala-Phe-Arg-OH 12 CEN-1 human nasopharyngeal carcinoma-targeting ligands
123B9 2225868-19-7 C58H82ClFN12O20 1321.79 {2-(3-chloro-4-fluorophenoxy)acetic acid}-SAYPDSVP-Nle-Hsr-S-NH2 {2-(3-chloro-4-fluorophenoxy)acetic acid}-Ser-Ala-Tyr-Pro-Asp-Ser-Val-Pro-Nle-Hsr-Ser-NH2 11 EphA2 agonist
C7 2159055-74-8 C62H90N18O16S1 1375.57 H2N-MHTAPGWGYRLS-OH H2N-Met-His-Thr-Ala-Pro-Gly-Trp-Gly-Tyr-Arg-Leu-Ser-OH 12 FRα-targeting peptide