ICI 154,129

Name: ICI 154,129
Brand: Creative Peptides
SKU: R1073
Availability: MadeToOrder

ICI 154129, a peptide analog, is a selective δ opioid antagonist.

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CAT No: R1073

CAS No: 83420-94-4

Synonyms/Alias: 83420-94-4;ICI 154129;ICI 154,129;ICI-154129;UNII-97BUE7NR2M;(2S)-2-[[(2S)-2-[2-[[2-[[(2S)-2-[bis(prop-2-enyl)amino]-3-(4-hydroxyphenyl)propanoyl]amino]acetyl]amino]ethylsulfanyl]-3-phenylpropanoyl]amino]-4-methylpentanoic acid;N,N-Bis(allyl)-tyr-gly-gly-psi-methylthio-phe-leu;M 154,129;M-154,129;97BUE7NR2M;N,N-Bis(allyl)-tyrosyl-glycyl-glycyl-psi-methylthio-phenylalanyl-leucine;DTXSID00232349;N,N-Di-2-propenyl-L-tyrosylglycyl-(alphaS)-alpha-((2-aminoethyl)thio)benzenepropanoyl-L-leucine;Glycinamide, N,N-di-2-propenyl-L-tyrosyl-N-(2-((2-((1-carboxy-3-methylbutyl)amino)-2-oxo-1-(phenylmethyl)ethyl)thio)ethyl)-, (S-(R*,R*))-;L-Leucine, N,N-di-2-propenyl-L-tyrosylglycyl-(alphaS)-alpha-((2-aminoethyl)thio)benzenepropanoyl-;M-154129;L-LEUCINE, N,N-DI-2-PROPEN-1-YL-L-TYROSYLGLYCYL-(.ALPHA.S)-.ALPHA.-((2-AMINOETHYL)THIO)BENZENEPROPANOYL-;SCHEMBL4405821;ICI154129;ICI 154129;M 154129;M154129;M-154129;DTXCID50154840;AKOS024458661;HY-101233;CS-0021020;Q27272001;((S)-2-((2-(2-((S)-2-(Diallylamino)-3-(4-hydroxyphenyl)propanamido)acetamido)ethyl)thio)-3-phenylpropanoyl)-L-leucine;L-LEUCINE, N,N-DI-2-PROPEN-1-YL-L-TYROSYLGLYCYL-(ALPHAS)-ALPHA-((2-AMINOETHYL)THIO)BENZENEPROPANOYL-;

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Specification Technical Data Publications Customer reviews and Q&A

M.F/Formula	C34H46N4O6S
M.W/Mr.	638.8
Sequence	YGFL(Modifications: Tyr-1 = N,N-diallyl-Tyr, Gly-2 - Phe-3 peptide bond replaced with Psi-(CH2S))
Labeling Target	Opioid Receptor
Appearance	Solid powder
Purity	>98% (or refer to the Certificate of Analysis)
Activity	Antagonist

Long-term Storage Conditions	Soluble in DMSO
Shipping Condition	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Short-term Storage Conditions	Dry, dark and at 0 - 4 °C
Solubility	-20 °C
InChI	InChI=1S/C34H46N4O6S/c1-5-17-38(18-6-2)29(21-26-12-14-27(39)15-13-26)32(41)36-23-31(40)35-16-19-45-30(22-25-10-8-7-9-11-25)33(42)37-28(34(43)44)20-24(3)4/h5-15,24,28-30,39H,1-2,16-23H2,3-4H3,(H,35,40)(H,36,41)(H,37,42)(H,43,44)/t28-,29-,30-/m0/s1
InChI Key	CZRZYRKTYLLLRL-DTXPUJKBSA-N
Isomeric SMILES	CC(C)C[C@@H](C(=O)O)NC(=O)[C@H](CC1=CC=CC=C1)SCCNC(=O)CNC(=O)[C@H](CC2=CC=C(C=C2)O)N(CC=C)CC=C
BoilingPoint	929.4ºC at 760 mmHg
ShelfLife	>3 years if stored properly
Melting Point	N/A

1. Effect of Short-Term Desiccation, Recovery Time, and CAPA-PVK Neuropeptide on the Immune System of the Burying Beetle Nicrophorus vespilloides

2. Identification, Localization in the Central Nervous System and Novel Myostimulatory Effect of Allatostatins in Tenebrio molitor Beetle

3. Glucagonlike peptide 2 analogue teduglutide: stimulation of proliferation but reduction of differentiation in human Caco-2 intestinal epithelial cells

4. Adipose tissue is a key organ for the beneficial effects of GLP-2 metabolic function

5. Novel Peptide-Based PD1 Immunomodulators Demonstrate Efficacy in Infectious Disease Vaccines and Therapeutics

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