Difelikefalin acetate

Difelikefalin ,also known as D-Phe-D-Phe-D-Leu-D-Lys-[γ-(4-N-piperidinyl)amino carboxylic acid] (as the acetate salt), is an analgesic opioid peptide acting as a peripherally specific, highly selective agonist of the κ-opioid receptor (KOR).

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CAT#10-101-174
CAS1024828-77-0(net);1024829-44-4
Synonyms/AliasCR845 acetate;CR-845 acetate;UNII-0P70AR5BYB; 0P70AR5BYB;
M.F/FormulaC38H57N7O8
M.W/Mr.739.90128
Labeling TargetK-opioid receptor
ApplicationDifelikefalin is an intravenous agent for the treatment of postoperative pain.
ActivityAgonist
Biological ActivityDifelikefalin acetate is a kappa opiate receptor agonist that is used for its antipruritic effects.
Areas of InterestPostoperative pain
DiseaseAcute Pain and Postoperative Pain
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