Potent and selective antagonist of bradykinin b1 receptor (pa2 = 8.49), which displays no activity at b2 receptors, and reduces mechanical hypernociception in a mouse model of neuropathic pain.
CAT# | R1087 |
CAS | 185052-09-9 |
M.F/Formula | C57H81N13O12 |
M.W/Mr. | 1140.35 |
Sequence | KRPPGFSXI(Modifications: Lys-1 = N-terminal Ac, X = DβNal) |
Labeling Target | Bradykinin Receptors |
Appearance | White lyophilised solid |
Purity | >98% |
Activity | Antagonist |
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