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Bestatin hydrochloride

Bestatin hydrochloride is a reversible inhibitor of aminopeptidase enzymes, namely Aminopeptidase B, Aminopeptidase M (CD13), and leucine aminopeptidase (LAP3). Inhibition of these proteins by bestatin correlates to apoptosis induction in oncogenic cells. Bestatin is also a potent inhibitor of leukotriene A4 hydrolase (LTA4). It is potentially used for cancer treatment.

Designed for biological research and industrial applications, not intended for individual clinical or medical purposes.

CAT No: R1028

CAS No:65391-42-6

Synonyms/Alias:Aminopeptidase inhibitor; leucine aminopeptidase; aminopeptidase B; NK-421

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M.F/Formula
C16H24N2O4 · HCl
M.W/Mr.
344.83
Labeling Target
Aminopeptidase
Appearance
White solid powder
Purity
>98% (or refer to the Certificate of Analysis)
Activity
Inhibitor
Long-term Storage Conditions
Soluble in DMSO
Shipping Condition
Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Short-term Storage Conditions
Dry, dark and at 0 - 4 °C
Solubility
-20 °C
InChI
InChI=1S/C16H24N2O4.ClH/c1-10(2)8-13(16(21)22)18-15(20)14(19)12(17)9-11-6-4-3-5-7-11;/h3-7,10,12-14,19H,8-9,17H2,1-2H3,(H,18,20)(H,21,22);1H/t12-,13+,14+;/m1./s1
InChI Key
XGDFITZJGKUSDK-UDYGKFQRSA-N
Isomeric SMILES
CC(C)C[C@@H](C(=O)O)NC(=O)[C@H]([C@@H](CC1=CC=CC=C1)N)O.Cl
BoilingPoint
604.7ºC at 760 mmHg
ShelfLife
>2 years if stored properly
Melting Point
216-218 °C

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