Urotensin-II (UT) receptor ligand that competitively antagonizes U-II induced contractions in the rat aorta (pIC50 = 7.46) and prevents plasma extravasation elicited by U-II in mice in vivo. Behaves as a silent antagonist in most in vitro assays and in vivo, but does retain small residual agonist activity under certain conditions in some assays.
CAT# | R1011 |
CAS | 879497-82-2 |
M.F/Formula | C50H64N10O12S2 |
M.W/Mr. | 1061.24 |
Sequence | H-Asp-DL-Pen(1)-Phe-D-Trp-DL-Dab-Tyr-Cys(1)-Val-OH |
Labeling Target | Urotensin-II receptor |
Appearance | White lyophilised solid |
Purity | >98% |
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