CYT-1010 is an μ-opioid receptor ligand potentially for the treatment of acute and chronic pain and neuropathic pain syndrome.
CAT# | 10-101-237 |
Chemical Structure | |
CAS | 213769-33-6 |
Synonyms/Alias | CYT1010, CYT 1010 |
Chemical Name | 2-amino-N-[3-benzyl-6-(1H-indol-3-ylmethyl)-2,5,8-trioxo-1,4,7-triazacyclotridec-9-yl]-3-(4-hydroxyphenyl)propanamide |
M.F/Formula | C35H40N6O5 |
M.W/Mr. | 624.73 |
Application | Acute and chronic pain and neuropathic pain syndrome |
Appearance | Solid powder |
Activity | Agonist |
Biological Activity | CYT-1010 is a mu-opioid receptor agonist extracted from patent WO2013173730A2, with EC50s of 13.1 nM and 0.0053 nM on beta-arrestin recruitment and inhibition of cAMP production, respectively. |
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